What is Butalbital and Where to Buy Butalbital ?

Butalbital, or 5-allyl-5-isobutylbarbituric acid, is a derivative of barbituric acid which the hydrogens at position 5 are substituted by an allyl group and an isobutyl group.

It is a short-to-intermediate acting member of barbiturates that exhibit muscle-relaxing and anti-anxiety properties that produce central nervous system (CNS) depression that ranges from mild sedation to general anesthesia 1. Butalbital has a low degree of selectivity and a narrow therapeutic index.

Typically indicated to manage tension (or muscle contraction) headaches, butalbital is often combined with one or more therapeutic agents, such as acetylsalicylic acid, acetaminophen, aspirin, and caffeine. There have not been clinical trials that evaluate the clinical efficacy of butalbital in migraines  thus it is not indicated for such condition.

As with other barbiturates, butalbital carries a risk of abuse or misuse potential, intoxication, hangover, tolerance, dependence, and over-dosage possibly leading to death Label.

Butalbital‐containing analgesics can also produce a drug‐induced headache in addition to tolerance and dependence. Due to these risks, the use of butalbital-containing combination products is typically limited for use only in cases where other medications are deemed ineffective and such usage is advised to be carefully monitored.

Buy Fioricet Online
Buy Fioricet Online

Butalbital, acetaminophen, and caffeine combination is used to relieve symptoms of tension (or muscle contraction) headaches.

Butalbital belongs to the group of medicines called barbiturates. Barbiturates act in the central nervous system (CNS) to produce their effects.

Fioricet is a prescription medication typically prescribed as a treatment for tension headaches. The medication is also available as an opiate painkiller, and experiencing a Fioricet withdrawal is a definite possibility when someone has taken the substance regularly for a long period of time.

When a person goes through the process of withdrawing from a substance, including prescription painkillers, it’s essentially the body going into shock. The individual may have been taking the substance for such a long period of time that their body and brain became used to the substance’s presence. When someone with Fioricet use disorder suddenly stops taking the substance, their body feels like it’s lost a sense of normalcy and balance.

The medical definition of withdrawal symptoms include anything that’s psychological or physically abnormal that occurs after an individual stops taking a substance to which they had a  physical dependence on. Similar to opioid withdrawal, some of the common Fioricet withdrawal symptoms include sweating, vomiting, and insomnia.

The withdrawal symptoms of any substance can range from being mildly uncomfortable to nearly debilitating, but the key to stopping substance misuse is going through withdrawal without too many complications. One of the best ways to do this for Fioricet, or any substance, is in a medically supervised detoxification program.

During a medically supervised detox, medical professionals and addiction specialists can help clients remain comfortable and then give them the tools and resources they need to begin on the path to recovery.

Acetaminophen is used to relieve pain and reduce fever in patients. It does not become habit-forming when taken for a long time. But acetaminophen may cause other unwanted effects when taken in large doses, including liver damage.

When butalbital is used for a long time, it may become habit-forming, causing mental or physical dependence. However, people who have continuing pain should not let the fear of dependence keep them from using narcotics to relieve their pain. Physical dependence may lead to withdrawal side effects if treatment is stopped suddenly. However, severe withdrawal side effects can usually be prevented by gradually reducing the dose over a period of time before treatment is stopped completely.

Caffeine is a CNS stimulant that is used with pain relievers to increase their effect. It has also been used for migraine headaches. However, caffeine can also cause physical dependence when it is used for a long time. This may lead to withdrawal (rebound) headaches when you stop taking it.

This medicine is available only with your doctor’s prescription.

Before taking this medicine

Do not use Fioricet if you have taken an MAO inhibitor in the past 14 days. A dangerous drug interaction could occur. MAO inhibitors include isocarboxazid, linezolid, phenelzine, rasagiline, selegiline, and tranylcypromine.

You should not use Fioricet if you are allergic to acetaminophen, butalbital, or caffeine, if you have porphyria, or if you have recently used alcohol, sedatives, tranquilizers, or other narcotic medications.

To make sure Fioricet is safe for you, tell your doctor if you have:

  • liver disease, cirrhosis, a history of alcoholism or drug addiction, or if you drink more than 3 alcoholic beverages per day;
  • kidney disease;
  • asthma, sleep apnea, or other breathing disorder;
  • stomach ulcer or bleeding;
  • a history of skin rash caused by any medication;
  • a history of mental illness or suicidal thoughts; or
  • if you use medicine to prevent blood clots.

It is not known whether Fioricet will harm an unborn baby. If you use butalbital while you are pregnant, your baby could become dependent on the drug. This can cause life-threatening withdrawal symptoms in the baby after it is born. Babies born dependent on habit-forming medicine may need medical treatment for several weeks. Tell your doctor if you are pregnant or plan to become pregnant.

This medicine can pass into breast milk and may harm a nursing baby. Tell your doctor if you are breast-feeding a baby.

What other drugs will affect Fioricet?

Taking this medicine with other drugs that make you sleepy or slow your breathing can cause dangerous or life-threatening side effects. Ask your doctor before taking Fioricet with a sleeping pill, narcotic pain medicine, muscle relaxer, or medicine for anxiety, depression, or seizures.

Other drugs may interact with acetaminophen, butalbital, and caffeine, including prescription and over-the-counter medicines, vitamins, and herbal products. Tell each of your health care providers about all medicines you use now and any medicine you start or stop using.

What is Fioricet Used For?

If you have ever experienced a migraine, you know the level of misery it can bring. Migraines go well beyond the pain or pressure of a typical headache, and they’re often accompanied by symptoms that can range to uncomfortable to scary. When you have a migraine doctors believe it’s something different from just a bad headache. Instead of being related to blood vessels, doctors believe that a lot of what causes migraines has to do with neurological things like brain chemicals.

With that being said, people who suffer from migraines often search for treatments that will work for them, and they also tend to have to go through several different medications before they get to one that will work for them.

One medication people sometimes consider is Fioricet, but doctors warn this should be a last resort for migraines, and there’s some debate over whether or not it works at all for migraine sufferers.

Is Fioricet Used As A Migraine Treatment?

In some cases, Fioricet may be used as a migraine treatment, but it’s not a first or even second choice among physicians. There are a few reasons. First, as was touched on above, Fioricet is primarily used for the treatment of tension headaches, which are very different from migraines. A lot of doctors feel that Fioricet doesn’t even necessarily work on migraine pain. There are a lot of other treatment options that are more specifically for the treatment of migraines, and they work in ways that are different from Fioricet.According to the FDA, Fioricet isn’t approved for the treatment of migraines at all. It may have some benefits for migraine sufferers in that it can provide them with a sense of physiological calmness because of how it works on the central nervous system, but there again are better ways to treat migraines.

Another reason Fioricet isn’t necessarily an ideal migraine treatment is because of the risks that come with it.

Butalbital is a substance that can be habit-forming, and the use of Fioricet has actually led to addiction problems and physical dependence for some of the people who use it. It may be a prescription medicine, but that certainly doesn’t mean it’s risk-free.

Another risk associated with the use of Fioricet is the potential for liver toxicity from acetaminophen. Acetaminophen taken in large doses can result in liver injury and failure, and it has to be taken carefully and only as prescribed.

So, to sum up, what is Fioricet used for? The FDA approves the use of this prescription medication for the treatment of tension headaches primarily, as well as something called a post-dural puncture headache, which can occur following something like anesthesia administered in the spine.

The FDA doesn’t approve Fioricet for the treatment of migraine headaches, both because it’s not the most effective available treatment option, and also because there are risks that come with the use of Fioricet including addiction, dependence and side effects like potential liver toxicity.

Can Fioricet Get You High?

NO. I do not think Fioricet can get you high.

One of the key active ingredients responsible for the so-called Fioricet high is butalbital.

butalbital
Butalbital is a barbiturate that’s considered short-to-intermediate acting, and it can relieve symptoms of anxiety, reduce pain, relax muscles and act as a sedative. There are many neuropsychological effects of butalbital, some of which aren’t clearly understood to this day.
The belief is that the Fioricet high is caused by the fact that butalbital can increase the inhibition neurotransmitters in the brain called GABA.
But by rxlist,  the barbiturate butalbital addict per day is usually about 1,500 mg. One pill of fioricet contains 40mg butalbital. if you are taking 1,500mg per day, you will take more than 30 tablet of fioricet which contain 9000mg acetaminophen. If you have taken more than 9000mg acetaminophen, you will die. The max dosage of acetaminophen per day is 3000mg.
Besides,  As tolerance to barbiturates develops, the amount needed to maintain the same level of intoxication increases; tolerance to a fatal dosage, however, does not increase more than twofold. As this occurs, the margin between an intoxication dosage and fatal dosage becomes smaller.
The lethal dose of a barbiturate is far less if alcohol is also ingested. Major withdrawal symptoms (convulsions and delirium) may occur within 16 hours and last up to 5 days after abrupt cessation of these drugs. Intensity of withdrawal symptoms gradually declines over a period of approximately 15 days. Treatment of barbiturate dependence consists of cautious and gradual withdrawal of the drug.
Barbiturate-dependent patients can be withdrawn by using a number of different withdrawal regimens. One method involves initiating treatment at the patient’s regular dosage level and gradually decreasing the daily dosage as tolerated by the patient.
Fioricet can reduce anxiety and some people with anxiety disorders may take it for this reason, although this is not what it’s approved for. There is the potential for Fioricet to decrease feelings of anxiety even when it’s taken at a normal dose, and this is because of the impact of butalbital on GABA. For some people, a Fioricet high is actually just equated with a reduction in anxiety.
Not everyone will associate the use of this drug with the Fioricet high. Some of the factors that determine whether or not a person will experience a Fioricet high can include the dosage they take and their tolerance. Newer users may be more likely to experience what they would describe as the Fioricet high. Other factors that could influence this include the specific formulation of the drug and whether or not other substances are taken with it. Some people may try to extract the butalbital from Fioricet and remove it from the caffeine and acetaminophen for a greater high.
This is not only drug abuse, but might not even achieve the effects the person is looking for. It’s important to realize that there can be serious and deadly consequences associated with trying to achieve a Fioricet high.
This can include addiction, adverse reactions, brain damage, emotional crashes, and overdose. Since Fioricet has acetaminophen, if people abuse it to get high they may also sustain liver damage or failure.

What is Fioricet side effects ?

Commonly reported side effects for Fioricet include:

  • Euphoria
  • Dizziness
  • Drowsiness
  • Intoxicated feeling
  • Light-headedness
  • Nausea
  • Vomiting
  • Sedation
  • Substance dependence
  • Shortness of breath
  • Abdominal pain

Fioricet is implicated as causing repeat headaches with over-use.

Fioricet Effects of Addiction

Abusing Fioricet or being addicted to it can be incredibly dangerous for multiple reasons. The first is because of the acetaminophen. Acetaminophen in amounts of more than 4000 mg a day can lead to liver damage and acute liver failure, particularly if it’s also combined with alcohol. Then, there’s the dangers of overdose and respiratory depression that can come with the butalbital in Fioricet.
It’s important only to use Fioricet as instructed by your physician to avoid these risks and also to lower your risk of becoming addicted to it. Some of the signs of Fioricet addiction include:
  • Being preoccupied with the use of Fioricet or always trying to find more of it.
  • Doctor shopping to get multiple prescriptions.
  • Taking it any way other than how your doctor instructs you or regularly taking it for recurring headaches.
  • Developing a tolerance to Fioricet is one of the first side effects of Firocet abuse. With tolerance, you have to take higher doses to get an effect. This can not only indicate a Fioricet abuse problem, but it also puts you at a higher risk of an overdose or liver failure.

If you are experiencing Fioricet effects that could indicate you have a problem, it’s important to speak with your doctor. It is possible to develop a tolerance for this drug, as was touched on above, so if you suddenly stop taking it you may experience withdrawal. Your physician or an addiction specialist can help you determine the best actions to take if you have an addiction to barbiturates like Fioricet.

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Fioricet Precautions

It is very important that your doctor check your progress while you or your child are taking this medicine. This will allow your doctor to see if the medicine is working properly and to decide if you should continue to take it.

This medicine may be habit-forming. If you or your child feel that the medicine is not working as well, do not use more than your prescribed dose. Call your doctor for instructions.

Check with your doctor right away if you or your child have pain or tenderness in the upper stomach, pale stools, dark urine, loss of appetite, nausea, unusual tiredness or weakness, or yellow eyes or skin. These could be symptoms of a serious liver problem.

Serious skin reactions can occur with this medicine. Check with your doctor right away if you have blistering, peeling, or loose skin, red skin lesions, severe acne or skin rash, sores or ulcers on the skin, or fever or chills while you are using this medicine.

This medicine may cause serious allergic reactions, including anaphylaxis. Anaphylaxis can be life-threatening and requires immediate medical attention. Call your doctor right away if you or your child have a rash, itching, hoarseness, trouble breathing, trouble swallowing, or any swelling of your hands, face, or mouth while you are using this medicine.

This medicine may make you dizzy or drowsy. Make sure you know how you react to this medicine before you drive, use machines, or do anything else that could be dangerous if you are dizzy or not alert.

This medicine will add to the effects of alcohol and other CNS depressants (medicines that can make you drowsy or less alert). Some examples of CNS depressants are antihistamines or medicine for allergies or colds, sedatives, tranquilizers, or sleeping medicine, other prescription pain medicine or narcotics, medicine for seizures or barbiturates, muscle relaxants, or anesthetics, including some dental anesthetics. Also, there may be a greater risk of liver damage if you drink three or more alcoholic beverages while you are taking acetaminophen. Do not drink alcoholic beverages, and check with your doctor before taking any of these medicines while you are using this medicine.

Before you have any medical tests, tell the medical doctor in charge that you or your child are taking this medicine. The results of some tests may be affected by this medicine.

Do not take other medicines unless they have been discussed with your doctor. This includes prescription or nonprescription (over-the-counter [OTC]) medicines and herbal or vitamin supplements.

Fioricet dosing information

Usual Adult Dose of Fioricet for Headache:

Acetaminophen 300 mg, butalbital 50 mg, and caffeine 40 mg:
1 or 2 capsule(s) orally every 4 hours as needed. Maximum daily dose: 6 doses.

Acetaminophen 325 mg, butalbital 50 mg, and caffeine 40 mg:
1 or 2 tablet(s), capsule(s), or tablespoonful(s) orally every 4 hours.
Maximum daily dose: 6 doses

Acetaminophen 500 mg, butalbital 50 mg, and caffeine 40 mg:
1 tablet or capsule orally every 4 hours.
Maximum daily dose: 6 doses

Acetaminophen 750 mg, butalbital 50 mg, and caffeine 40 mg:
1 tablet orally every 4 hours.
Maximum daily dose: 5 tablets

Usual Pediatric Dose of Fioricet for Headache:

12 years and older:
Acetaminophen 300 mg, butalbital 50 mg, and caffeine 40 mg:
1 or 2 capsule(s) orally every 4 hours as needed. Maximum daily dose: 6 doses.

What should I know before I take Fioricet ?

Do not use Fioricet if you have taken an MAO inhibitor in the past 14 days. A dangerous drug interaction could occur. MAO inhibitors include isocarboxazid, linezolid, phenelzine, rasagiline, selegiline, and tranylcypromine.

You should not use Fioricet if you are allergic to acetaminophen, butalbital, or caffeine, if you have porphyria, or if you have recently used alcohol, sedatives, tranquilizers, or other narcotic medications.

To make sure Fioricet is safe for you, tell your doctor if you have:

  • liver disease, cirrhosis, a history of alcoholism or drug addiction, or if you drink more than 3 alcoholic beverages per day;
  • kidney disease;
  • asthma, sleep apnea, or other breathing disorder;
  • stomach ulcer or bleeding;
  • a history of skin rash caused by any medication;
  • a history of mental illness or suicidal thoughts; or
  • if you use medicine to prevent blood clots.

It is not known whether Fioricet will harm an unborn baby. If you use butalbital while you are pregnant, your baby could become dependent on the drug. This can cause life-threatening withdrawal symptoms in the baby after it is born. Babies born dependent on habit-forming medicine may need medical treatment for several weeks. Tell your doctor if you are pregnant or plan to become pregnant.

This medicine can pass into breast milk and may harm a nursing baby. Tell your doctor if you are breast-feeding a baby.